De Luca V.; Angeli A.; Mazzone V.; Adelfio C.; Carginale V.; Scaloni A.; Carta F.; Selleri S.; Supuran C.T.; Capasso C. (2022). Heterologous expression and biochemical characterisation of the recombinant β-carbonic anhydrase (MpaCA) from the warm-blooded vertebrate pathogen malassezia pachydermatis. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 37, pp. 62-68, ISSN:1475-6366 DOI  

  Giovannuzzi S.; Abutaleb N.S.; Hewitt C.S.; Carta F.; Nocentini A.; Seleem M.N.; Flaherty D.P.; Supuran C.T. (2022). Dithiocarbamates effectively inhibit the α-carbonic anhydrase from Neisseria gonorrhoeae. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 37, pp. 1-8, ISSN:1475-6366 DOI  

  Testa, Chiara; Papini, Anna Maria; Zeidler, Reinhard; Vullo, Daniela; Carta, Fabrizio; Supuran, Claudiu T; Rovero, Paolo (2022). First studies on tumor associated carbonic anhydrases IX and XII monoclonal antibodies conjugated to small molecule inhibitors. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 37, pp. 592-596, ISSN:1475-6366 DOI  

  Akgul O.; Lucarini E.; Mannelli L.D.C.; Ghelardini C.; D'Ambrosio K.; Buonanno M.; Monti S.M.; De Simone G.; Angeli A.; Supuran C.T.; Carta F. (2022). Sultam based Carbonic Anhydrase VII inhibitors for the management of neuropathic pain. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 227, pp. 0-0, ISSN:0223-5234 DOI  

  Angeli A.; Velluzzi A.; Selleri S.; Capasso C.; Spadini C.; Iannarelli M.; Cabassi C.S.; Carta F.; Supuran C.T. (2022). Seleno Containing Compounds as Potent and Selective Antifungal Agents. ACS INFECTIOUS DISEASES, vol. 8, pp. 1905-1919, ISSN:2373-8227 DOI  

  Eysteinsson T.; Garcia-Llorca A.; Angeli A.; Supuran C.T.; Carta F. (2022). Vasodilation of Pre-contracted Porcine Retinal Arteries by Carbonic Anhydrase Inhibitors with Enhanced Lipophilicity. CURRENT EYE RESEARCH, vol. 47, pp. 1615-1621, ISSN:0271-3683 DOI  

  Liguori F.; Carradori S.; Ronca R.; Rezzola S.; Filiberti S.; Carta F.; Turati M.; Supuran C.T. (2022). Benzenesulfonamides with different rigidity-conferring linkers as carbonic anhydrase inhibitors: an insight into the antiproliferative effect on glioblastoma, pancreatic, and breast cancer cells. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 37, pp. 1857-1869, ISSN:1475-6366 DOI  

  Angeli A.; Ferraroni M.; Carta F.; Haberli C.; Keiser J.; Costantino G.; Supuran C.T. (2022). Development of Praziquantel sulphonamide derivatives as antischistosomal drugs. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 37, pp. 1479-1494, ISSN:1475-6366 DOI  

  Bozdag M.; Cravey L.; Combs J.; Kota A.; McKenna R.; Angeli A.; Selleri S.; Carta F.; Supuran C.T. (2022). Small Molecule Alkoxy Oriented Selectiveness on Human Carbonic Anhydrase II and IX Inhibition. CHEMMEDCHEM, vol. 17, pp. 0-0, ISSN:1860-7179 DOI  

  Gumus A.; Bozdag M.; Akdemir A.; Angeli A.; Selleri S.; Carta F.; Supuran C.T. (2022). Thiosemicarbazide-Substituted Coumarins as Selective Inhibitors of the Tumor Associated Human Carbonic Anhydrases IX and XII. MOLECULES, vol. 27, pp. 0-0, ISSN:1420-3049 DOI  

  Emanuela Berrino; Bastien Michelet; Agnes Martin-Mingot; Fabrizio Carta; Claudiu Supuran; Sebastien Thibaudeau (2021). Modulating the Efficacy of Carbonic Anhydrase Inhibitors through Fluorine Substitution. ANGEWANDTE CHEMIE. INTERNATIONAL EDITION, pp. 0-0, ISSN:1433-7851 DOI  

  Angeli A.; Berrino E.; Carradori S.; Supuran C.T.; Cirri M.; Carta F.; Costantino G. (2021). Amine-and amino acid-based compounds as carbonic anhydrase activators. MOLECULES, vol. 26, pp. 0-0, ISSN:1420-3049 DOI  

  Berrino E.; Carradori S.; Angeli A.; Carta F.; Supuran C.T.; Guglielmi P.; Coletti C.; Paciotti R.; Schweikl H.; Maestrelli F.; Cerbai E.; Gallorini M. (2021). Dual carbonic anhydrase ix/xii inhibitors and carbon monoxide releasing molecules modulate LPS-mediated inflammation in mouse macrophages. ANTIOXIDANTS, vol. 10, pp. 1-24, ISSN:2076-3921 DOI  

  Tanini D.; Carradori S.; Capperucci A.; Lupori L.; Zara S.; Ferraroni M.; Ghelardini C.; Mannelli L.D.C.; Micheli L.; Lucarini E.; Carta F.; Angeli A.; Supuran C.T. (2021). Chalcogenides-incorporating carbonic anhydrase inhibitors concomitantly reverted oxaliplatin-induced neuropathy and enhanced antiproliferative action. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 225, pp. 0-0, ISSN:0223-5234 DOI  

  Chen F.; Licarete E.; Wu X.; Petrusca D.; Maguire C.; Jacobsen M.; Colter A.; Sandusky G.E.; Czader M.; Capitano M.L.; Ropa J.P.; Boswell H.S.; Carta F.; Supuran C.T.; Parkin B.; Fishel M.L.; Konig H. (2021). Pharmacological inhibition of Carbonic Anhydrase IX and XII to enhance targeting of acute myeloid leukaemia cells under hypoxic conditions. JOURNAL OF CELLULAR AND MOLECULAR MEDICINE, vol. 25, pp. 11039-11052, ISSN:1582-1838 DOI  

  Vaiano F.; Bertol E.; Mineo M.; Pietrosemoli L.; Rubicondo J.; Supuran C.T.; Carta F. (2021). Development of a new lc-ms/ms screening method for detection of 120 nps and 43 drugs in blood. SEPARATIONS, vol. 8, pp. 0-0, ISSN:2297-8739 DOI  

  De Luca V.; Angeli A.; Mazzone V.; Adelfio C.; Carta F.; Selleri S.; Carginale V.; Scaloni A.; Supuran C.T.; Capasso C. (2021). Inhibitory effects of sulfonamide derivatives on the β‐carbonic anhydrase (Mpaca) from malassezia pachydermatis, a commensal, pathogenic fungus present in domestic animals. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, vol. 22, pp. 0-0, ISSN:1661-6596 DOI  

  Chafe, Shawn C; Vizeacoumar, Frederick S; Venkateswaran, Geetha; Nemirovsky, Oksana; Awrey, Shannon; Brown, Wells S; McDonald, Paul C; Carta, Fabrizio; Metcalfe, Andrew; Karasinska, Joanna M; Huang, Ling; Muthuswamy, Senthil K; Schaeffer, David F; Renouf, Daniel J; Supuran, Claudiu T; Vizeacoumar, Franco J; Dedhar, Shoukat (2021). Genome-wide synthetic lethal screen unveils novel CAIX-NFS1/xCT axis as a targetable vulnerability in hypoxic solid tumors. SCIENCE ADVANCES, vol. 7, pp. 0-0, ISSN:2375-2548 DOI  

  Andrea Angeli; Marta Ferraroni; Akram A. Da’dara; Silvia Selleri; Mariana Pinteala; Fabrizio Carta; Patrick J. Skelly; Claudiu T. Supuran (2021). Structural Insights into Schistosoma mansoni Carbonic Anhydrase (SmCA) Inhibition by Selenoureido-Substituted Benzenesulfonamides. JOURNAL OF MEDICINAL CHEMISTRY, pp. 0-0, ISSN:0022-2623 DOI  

  Marialucia Gallorini; Anna C. Berardi; Alessia Ricci; Cristina Antonetti Lamorgese Passeri; Susi Zara; Francesco Oliva; Amelia Cataldi; Fabrizio Carta; Simone Carradori (2021). Dual Acting Carbon Monoxide Releasing Molecules and Carbonic Anhydrase Inhibitors Differentially Modulate Inflammation in Human Tenocytes. BIOMEDICINES, vol. 9, pp. 0-0, ISSN:2227-9059 DOI  

  Lenci E.; Angeli A.; Calugi L.; Innocenti R.; Carta F.; Supuran C.T.; Trabocchi A. (2021). Multitargeting application of proline-derived peptidomimetics addressing cancer-related human matrix metalloproteinase 9 and carbonic anhydrase II. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 214, pp. 0-0, ISSN:0223-5234 DOI  

  Plyasova A.A.; Berrino E.; Khan I.I.; Veselovsky A.V.; Pokrovsky V.S.; Angeli A.; Ferraroni M.; Supuran C.T.; Pokrovskaya M.V.; Alexandrova S.S.; Gladilina Y.A.; Sokolov N.N.; Hilal A.; Carta F.; Zhdanov D.D. (2021). Mechanisms of the Antiproliferative and Antitumor Activity of Novel Telomerase-Carbonic Anhydrase Dual-Hybrid Inhibitors. JOURNAL OF MEDICINAL CHEMISTRY, vol. 64, pp. 11432-11444, ISSN:0022-2623 DOI  

  Sethi K.K.; Mishra K.M.A.; Verma S.M.; Vullo D.; Carta F.; Supuran C.T. (2021). Synthesis and human carbonic anhydrase I, II, IX, and XII inhibition studies of sulphonamides incorporating mono-, Bi- and tricyclic imide moieties. PHARMACEUTICALS, vol. 14, pp. 0-0, ISSN:1424-8247 DOI  

  Gumus A.; Bozdag M.; Angeli A.; Peat T.S.; Carta F.; Supuran C.T.; Selleri S. (2021). Privileged scaffolds in medicinal chemistry: Studies on pyrazolo[1,5-a]pyrimidines on sulfonamide containing Carbonic Anhydrase inhibitors. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 49, pp. 0-0, ISSN:0960-894X DOI  

  Nocentini, Alessio; Angeli, Andrea; Carta, Fabrizio; Winum, Jean-Yves; Zalubovskis, Raivis; Carradori, Simone; Capasso, Clemente; Donald, William A; Supuran, Claudiu T (2021). Reconsidering anion inhibitors in the general context of drug design studies of modulators of activity of the classical enzyme carbonic anhydrase. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 36, pp. 561-580, ISSN:1475-6366 DOI  

  Akgul O.; Angeli A.; Selleri S.; Capasso C.; Supuran C.T.; Carta F. (2021). Taurultams incorporating arylsulfonamide: First in vitro inhibition studies of α-, β- and γ-class Carbonic Anhydrases from Vibrio cholerae and Burkholderia pseudomallei. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 219, pp. 0-0, ISSN:0223-5234 DOI  

  Angeli A.; Pinteala M.; Maier S.S.; Toti A.; Di Cesare Mannelli L.; Ghelardini C.; Selleri S.; Carta F.; Supuran C.T. (2021). Tellurides bearing benzensulfonamide as carbonic anhydrase inhibitors with potent antitumor activity. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 45, pp. 0-0, ISSN:0960-894X DOI  

  Debora Pratesi, Andrea Sodini, Camilla Matassini, Francesca Cardona, Andrea Angeli, Fabrizio Carta, Marta Ferraroni, Claudiu T. Supuran, Andrea Goti (2021). Synthesis of Azasugar–Sulfonamide conjugates and their Evaluation as Inhibitors of Carbonic Anhydrases: the Azasugar Approach to Selectivity. EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, vol. 2021, pp. 2604-2614, ISSN:1099-0690 DOI  

  Mansoldo F.R.P.; Berrino E.; Guglielmi P.; Carradori S.; Carta F.; Secci D.; Supuran C.T.; Vermelho A.B. (2021). An innovative spectroscopic approach for qualitative and quantitative evaluation of Mb-CO from myoglobin carbonylation reaction through chemometrics methods. SPECTROCHIMICA ACTA. PART A, MOLECULAR AND BIOMOLECULAR SPECTROSCOPY, pp. 0-0, ISSN:1386-1425 DOI  

  Vannozzi G.; Vullo D.; Angeli A.; Ferraroni M.; Combs J.; Lomelino C.; Andring J.; Mckenna R.; Bartolucci G.; Pallecchi M.; Lucarini L.; Sgambellone S.; Masini E.; Carta F.; Supuran C.T. (2021). One-Pot Procedure for the Synthesis of Asymmetric Substituted Ureido Benzene Sulfonamides as Effective Inhibitors of Carbonic Anhydrase Enzymes. JOURNAL OF MEDICINAL CHEMISTRY, vol. 65, pp. 824-837-837, ISSN:0022-2623 DOI  

  Angeli A.; Carta F.; Nocentini A.; Winum J.-Y.; Zalubovskis R.; Onnis V.; Eldehna W.M.; Capasso C.; Carradori S.; Donald W.A.; Dedhar S.; Supuran C.T. (2021). Response to Perspectives on the Classical Enzyme Carbonic Anhydrase and the Search for Inhibitors. BIOPHYSICAL JOURNAL, vol. 120, pp. 178-181, ISSN:0006-3495 DOI  

  Aspatwar, Ashok; Hammaren, Milka; Parikka, Mataleena; Parkkila, Seppo; Carta, Fabrizio; Bozdag, Murat; Vullo, Daniela; Supuran, Claudiu T (2020). In vitro inhibition of Mycobacterium tuberculosis β-carbonic anhydrase 3 with Mono- and dithiocarbamates and evaluation of their toxicity using zebrafish developing embryos. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 35, pp. 65-71-71, ISSN:1475-6366 DOI  

  Pratesi, Debora; Matassini, Camilla; Goti, Andrea; Angeli, Andrea; Carta, Fabrizio; Supuran, Claudiu T.; Spanevello, Rolando; Cardona, Francesca (2020). Glycomimetic Based Approach toward Selective Carbonic Anhydrase Inhibitors. ACS MEDICINAL CHEMISTRY LETTERS, vol. 11, pp. 727-731, ISSN:1948-5875 DOI  

  Berrino E.; Angeli A.; Zhdanov D.D.; Kiryukhina A.P.; Milaneschi A.; De Luca A.; Bozdag M.; Carradori S.; Selleri S.; Bartolucci G.; Peat T.S.; Ferraroni M.; Supuran C.T.; Carta F. (2020). Azidothymidine "clicked" into 1,2,3-Triazoles: First Report on Carbonic Anhydrase-Telomerase Dual-Hybrid Inhibitors. JOURNAL OF MEDICINAL CHEMISTRY, vol. 63, pp. 7392-7409, ISSN:0022-2623 DOI  

  Angeli A.; Peat T.S.; Selleri S.; Saleh Alfawaz Altamimi A.; Supuran C.T.; Carta F. (2020). X-ray crystallography of Epacadostat in adduct with Carbonic Anhydrase IX. BIOORGANIC CHEMISTRY, vol. 97, pp. 103669-103669, ISSN:0045-2068 DOI  

  Scheila Daiane Schmidt, Alessia Costa, Barbara Rani, Eduarda Godfried Nachtigall, Maria Beatrice Passani, Fabrizio Carta, Alessio Nocentini, Jociane de Carvalho Myskiw, Cristiane Regina Guerino Furini, Claudiu T. Supuran, Ivan Izquierdo, Patrizio Blandina, Gustavo Provensi (2020). The role of carbonic anhydrases in extinction of contextual fear memory. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, pp. 1-9, ISSN:0027-8424 DOI  

  Angeli, Andrea; Carta, Fabrizio; Donnini, Selene; Capperucci, Antonella; Ferraroni, Marta; Tanini, Damiano; Supuran, Claudiu T (2020). Selenolesterase enzyme activity of carbonic anhydrases. CHEMICAL COMMUNICATIONS, pp. 0-0, ISSN:1359-7345 DOI  

  Angeli, Andrea; Etxebeste-Mitxeltorena, Mikel; Sanmartín, Carmen; Espuelas, Socorro; Moreno, Esther; Azqueta, Amaya; Parkkila, Seppo; Carta, Fabrizio; Supuran, Claudiu T (2020). Tellurides Bearing Sulfonamides as Novel Inhibitors of Leishmanial Carbonic Anhydrase with Potent Antileishmanial Activity. JOURNAL OF MEDICINAL CHEMISTRY, pp. 0-0, ISSN:0022-2623 DOI  

  Ali, Majid; Bozdag, Murat; Farooq, Umar; Angeli, Andrea; Carta, Fabrizio; Berto, Paola; Zanotti, Giuseppe; Supuran, Claudiu T (2020). Benzylaminoethyureido-Tailed Benzenesulfonamides: Design, Synthesis, Kinetic and X-ray Investigations on Human Carbonic Anhydrases. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, vol. 21, pp. 2560-2560, ISSN:1422-0067 DOI  

  Ruzzolini J, Laurenzana A, Andreucci E, Peppicelli S, Bianchini F, Carta F, Supuran CT, Romanelli MN, Nediani C, Calorini L. (2020). A potentiated cooperation of carbonic anhydrase IX and histone deacetylase inhibitors against cancer. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 35, pp. 391-397, ISSN:1475-6366 DOI  

  Emanuela Berrino, Claudiu Supuran, Alessandro Mugelli, Fabrizio Carta (2020). Carbonic Anhydrase Inhibitors: Versatile Agents for the Treatment of Human Diseases. (Tutor: Claudiu Supuran, Alessandro Mugelli)

  Bua S.; Lucarini L.; Micheli L.; Menicatti M.; Bartolucci G.; Selleri S.; Di Cesare Mannelli L.; Ghelardini C.; Masini E.; Carta F.; Gratteri P.; Nocentini A.; Supuran C.T. (2020). Bioisosteric Development of Multitarget Nonsteroidal Anti-Inflammatory Drug-Carbonic Anhydrases Inhibitor Hybrids for the Management of Rheumatoid Arthritis. JOURNAL OF MEDICINAL CHEMISTRY, vol. 63, pp. 2325-2342, ISSN:0022-2623 DOI   Accesso ONLINE all'editore

  Angeli, Andrea; Pinteala, Mariana; Maier, Stelian S; Simionescu, Bogdan C; Milaneschi, Andrea; Abbas, Ghulam; Del Prete, Sonia; Capasso, Clemente; Capperucci, Antonella; Tanini, Damiano; Carta, Fabrizio; Supuran, Claudiu T (2020). Evaluation of Thio- and Seleno-Acetamides Bearing Benzenesulfonamide as Inhibitor of Carbonic Anhydrases from Different Pathogenic Bacteria. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, vol. 21, pp. 598-598, ISSN:1422-0067 DOI  

  Bozdag M.; Supuran C.T.; Esposito D.; Angeli A.; Carta F.; Monti S.M.; De Simone G.; Alterio V. (2020). 2-Mercaptobenzoxazoles: a class of carbonic anhydrase inhibitors with a novel binding mode to the enzyme active site. CHEMICAL COMMUNICATIONS, vol. 56, pp. 8297-8300, ISSN:1359-7345 DOI  

  Akgul O.; Angeli A.; Vullo D.; Carta F.; Supuran C.T. (2020). Unconventional amino acids in medicinal chemistry: First report on taurine merged within carbonic anhydrase inhibitors. BIOORGANIC CHEMISTRY, vol. 103, pp. 0-0, ISSN:0045-2068 DOI  

  Clima L.; Craciun B.F.; Angeli A.; Petreni A.; Bonardi A.; Nocentini A.; Carta F.; Gratteri P.; Pinteala M.; Supuran C.T. (2020). Synthesis, Computational Studies and Assessment of in Vitro Activity of Squalene Derivatives as Carbonic Anhydrase Inhibitors. CHEMMEDCHEM, vol. 15, pp. 2052-2057, ISSN:1860-7179 DOI  

  Aspatwar A.; Berrino E.; Bua S.; Carta F.; Capasso C.; Parkkila S.; Supuran C.T. (2020). Toxicity evaluation of sulfamides and coumarins that efficiently inhibit human carbonic anhydrases. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 35, pp. 1765-1772, ISSN:1475-6366 DOI  

  Angeli A.; Carta F.; Nocentini A.; Winum J.-Y.; Zalubovskis R.; Akdemir A.; Onnis V.; Eldehna W.M.; Capasso C.; Simone G.D.; Monti S.M.; Carradori S.; Donald W.A.; Dedhar S.; Supuran C.T. (2020). Carbonic anhydrase inhibitors targeting metabolism and tumor microenvironment. METABOLITES, vol. 10, pp. 1-21, ISSN:2218-1989 DOI  

  Mori M.; Capasso C.; Carta F.; Donald W.A.; Supuran C.T. (2020). A deadly spillover: SARS-CoV-2 outbreak. EXPERT OPINION ON THERAPEUTIC PATENTS, vol. 30, pp. 481-485, ISSN:1354-3776 DOI  

  Ali M.; Angeli A.; Bozdag M.; Carta F.; Capasso C.; Farooq U.; Supuran C.T. (2020). Benzylaminoethylureido-Tailed Benzenesulfonamides Show Potent Inhibitory Activity against Bacterial Carbonic Anhydrases. CHEMMEDCHEM, pp. 0-0, ISSN:1860-7179 DOI  

  Angeli A.; Carta F.; Supuran C.T. (2020). Carbonic anhydrases: Versatile and useful biocatalysts in chemistry and biochemistry. CATALYSTS, vol. 10, pp. 1-11, ISSN:2073-4344 DOI  

  Poli G.; Bozdag M.; Berrino E.; Angeli A.; Tuccinardi T.; Carta F.; Supuran C.T. (2020). N-aryl-N′-ureido-O-sulfamates as potent and selective inhibitors of hCA VB over hCA VA: Deciphering the binding mode of new potential agents in mitochondrial dysfunctions. BIOORGANIC CHEMISTRY, vol. 100, pp. 0-0, ISSN:0045-2068 DOI  

  Costa G.; Maruca A.; Rocca R.; Ambrosio F.A.; Berrino E.; Carta F.; Mesiti F.; Salatino A.; Lanzillotta D.; Trapasso F.; Artese A.; Alcaro S.; Supuran C.T. (2020). In silico identification and biological evaluation of antioxidant food components endowed with IX and XII hCA inhibition. ANTIOXIDANTS, vol. 9, pp. 1-13, ISSN:2076-3921 DOI  

  Lucarini L.; Durante M.; Sgambellone S.; Lanzi C.; Bigagli E.; Akgul O.; Masini E.; Supuran C.T.; Carta F. (2020). Effects of new nsaid-cai hybrid compounds in inflammation and lung fibrosis. BIOMOLECULES, vol. 10, pp. 1-20, ISSN:2218-273X DOI  

  Felipe Raposo Passos Mansoldo; Fabrizio Carta; Andrea Angeli; Veronica da Silva Cardoso; Claudiu T. Supuran; Alane Beatriz Vermelho (2020). Chagas Disease: Perspectives on the Past and Present and Challenges in Drug Discovery. MOLECULES, vol. 25, pp. 0-0, ISSN:1420-3049 DOI  

  Akgul O.; Singh S.; Andring J.T.; McKenna R.; Selleri S.; Carta F.; Angeli A.; Supuran C.T. (2020). Handling drug-target selectivity: A study on ureido containing Carbonic Anhydrase inhibitors. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, pp. 0-0, ISSN:0223-5234 DOI  

  Angeli A.; Ferraroni M.; Pinteala M.; Maier S.S.; Simionescu B.C.; Carta F.; Del Prete S.; Capasso C.; Supuran C.T. (2020). Crystal structure of a tetrameric type II β-carbonic anhydrase from the pathogenic bacterium burkholderia pseudomallei. MOLECULES, vol. 25, pp. 2269-2278, ISSN:1420-3049 DOI  

  Andreucci, Elena; Ruzzolini, Jessica; Peppicelli, Silvia; Bianchini, Francesca; Laurenzana, Anna; Carta, Fabrizio; Supuran, Claudiu T.; Calorini, Lido (2019). The carbonic anhydrase IX inhibitor SLC-0111 sensitises cancer cells to conventional chemotherapy. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 34, pp. 117-123, ISSN:1475-6366 DOI   Accesso ONLINE all'editore

  Vullo D.; Carta F. (2019). Mechanisms of action of carbonic anhydrase inhibitors: Zinc binders. In: Claudiu T. Supuran, Alessio Nocentini. Carbonic Anhydrases Biochemistry and Pharmacology of an Evergreen Pharmaceutical Target, pp. 187-222 Elsevier, ISBN:978-0-12-816476-1. DOI  

  Bozdag M.; Poli G.; Angeli A.; Lucarini E.; Tuccinardi T.; Di Cesare Mannelli L.; Selleri S.; Ghelardini C.; Winum J.-Y.; Carta F.; Supuran C.T. (2019). N-aryl-N’-ureido-O-sulfamates: Potent and selective inhibitors of the human Carbonic Anhydrase VII isoform with neuropathic pain relieving properties. BIOORGANIC CHEMISTRY, vol. 89, pp. 103033-103043, ISSN:0045-2068 DOI   Accesso ONLINE all'editore

  Tanini, Damiano; Ricci, Lorenzo; Capperucci, Antonella; Di Cesare Mannelli, Lorenzo; Ghelardini, Carla; Peat, Thomas S; Carta, Fabrizio; Angeli, Andrea; Supuran, Claudiu T (2019). Synthesis of novel tellurides bearing benzensulfonamide moiety as carbonic anhydrase inhibitors with antitumor activity. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 181, pp. 111586-111594, ISSN:1768-3254 DOI  

  Bozdag, Murat; Ferraroni, Marta; Ward, Carol; Carta, Fabrizio; Bua, Silvia; Angeli, Andrea; Langdon, Simon P; Kunkler, Ian H; Al-Tamimi, Abdul-Malek S; Supuran, Claudiu T (2019). Carbonic anhydrase inhibitors based on sorafenib scaffold: Design, synthesis, crystallographic investigation and effects on primary breast cancer cells. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 182, pp. 111600-111611, ISSN:1768-3254 DOI  

  Al-Tamimi A.-M.S.; Etxebeste-Mitxeltorena M.; Sanmartin C.; Jimenez-Ruiz A.; Syrjanen L.; Parkkila S.; Selleri S.; Carta F.; Angeli A.; Supuran C.T. (2019). Discovery of new organoselenium compounds as antileishmanial agents. BIOORGANIC CHEMISTRY, vol. 86, pp. 339-345, ISSN:0045-2068 DOI   Accesso ONLINE all'editore

  Eysteinsson T.; Gudmundsdottir H.; Hardarson A.O.; Berrino E.; Selleri S.; Supuran C.T.; Carta F. (2019). Carbonic anhydrase inhibitors of different structures dilate pre-contracted porcine retinal arteries. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, vol. 20, pp. 467-479, ISSN:1661-6596 DOI   Accesso ONLINE all'editore

  Bozdag, Murat; Altamimi, Abdulmalik Saleh Alfawaz; Vullo, Daniela; Supuran, Claudiu T; Carta, Fabrizio (2019). State of the Art on Carbonic Anhydrase Modulators for Biomedical Purposes. CURRENT MEDICINAL CHEMISTRY, vol. 26, pp. 2558-2573, ISSN:0929-8673 DOI  

  Mboge M.Y.; Chen Z.; Khokhar D.; Wolff A.; Ai L.; Heldermon C.D.; Bozdag M.; Carta F.; Supuran C.T.; Brown K.D.; McKenna R.; Frost C.J.; Frost S.C. (2019). A non-catalytic function of carbonic anhydrase IX contributes to the glycolytic phenotype and pH regulation in human breast cancer cells. BIOCHEMICAL JOURNAL, vol. 476, pp. 1497-1513, ISSN:0264-6021 DOI   Accesso ONLINE all'editore

  Micheli L.; Bozdag M.; Akgul O.; Carta F.; Guccione C.; Bergonzi M.C.; Bilia A.R.; Cinci L.; Lucarini E.; Parisio C.; Supuran C.T.; Ghelardini C.; Di Cesare Mannelli L. (2019). Pain relieving effect of-NSAIDS-CAIs hybrid molecules: Systemic and intra-articular treatments against rheumatoid arthritis. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, vol. 20, pp. 1923-1938, ISSN:1422-0067 DOI   Accesso ONLINE all'editore

  Angeli A.; Di Cesare Mannelli L.; Ghelardini C.; Peat T.S.; Bartolucci G.; Menicatti M.; Carta F.; Supuran C.T. (2019). Benzensulfonamides bearing spyrohydantoin moieties act as potent inhibitors of human carbonic anhydrases II and VII and show neuropathic pain attenuating effects. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 177, pp. 188-197, ISSN:1768-3254 DOI   Accesso ONLINE all'editore

  Costa G.; Carta F.; Ambrosio F.A.; Artese A.; Ortuso F.; Moraca F.; Rocca R.; Romeo I.; Lupia A.; Maruca A.; Bagetta D.; Catalano R.; Vullo D.; Alcaro S.; Supuran C.T. (2019). A computer-assisted discovery of novel potential anti-obesity compounds as selective carbonic anhydrase VA inhibitors. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 181, pp. 111565-111572, ISSN:1768-3254 DOI  

  Berrino E.; Milazzo L.; Micheli L.; Vullo D.; Angeli A.; Bozdag M.; Nocentini A.; Menicatti M.; Bartolucci G.; Di Cesare Mannelli L.; Ghelardini C.; Supuran C.T.; Carta F. (2019). Synthesis and evaluation of carbonic anhydrase inhibitors with carbon monoxide releasing properties for the management of rheumatoid arthritis. JOURNAL OF MEDICINAL CHEMISTRY, vol. 62, pp. 7233-7249, ISSN:1520-4804 DOI  

  Laura Micheli, Murat Bozdag , Ozlem Akgul , Fabrizio Carta , Clizia Guccione, Maria Camilla Bergonzi, Anna Rita Bilia, Lorenzo Cinci, Elena Lucarini, Carmen Parisio, Claudiu T. Supuran , Carla Ghelardini, Lorenzo Di Cesare Mannelli (2019). Pain Relieving Eect of-NSAIDs-CAIs Hybrid Molecules: Systemic and Intra-Articular Treatments against Rheumatoid Arthritis. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, pp. 0-0, ISSN:1422-0067

  Carta, Fabrizio; Dumy, Pascal; Supuran, Claudiu T; Winum, Jean-Yves (2019). Multivalent Carbonic Anhydrases Inhibitors. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, vol. 20, pp. 5352-5367, ISSN:1422-0067 DOI  

  Kalisha Vali Y.; Gundla R.; Singh O.V.; Tamboli Y.; Di Cesare Manelli L.; Ghelardini C.; Al-Tamimi A.-M.S.; Carta F.; Angeli A.; Supuran C.T. (2019). Spirocyclic sulfonamides with carbonic anhydrase inhibitory and anti-neuropathic pain activity. BIOORGANIC CHEMISTRY, vol. 92, pp. 103210-103220, ISSN:0045-2068 DOI   Accesso ONLINE all'editore

  Tanini, Damiano; Capperucci, Antonella; Ferraroni, Marta; Carta, Fabrizio; Angeli, Andrea; Supuran, Claudiu T. (2019). Direct and Straightforward access to substituted alkyl selenols as novel carbonic anhydrase inhibitors. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, pp. 111811-111817, ISSN:0223-5234 DOI  

  Gustavo Provensi, Fabrizio Carta, Alessio Nocentini, Claudiu T. Supuran, Fiorella Casamenti, Maria Beatrice Passani, Silvia Fossati (2019). A New Kid on the Block? Carbonic Anhydrases as Possible New Targets in Alzheimer's Disease. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, vol. 20, pp. 4724-4741, ISSN:1422-0067 DOI  

  Berrino E.; Carta F. (2019). Carbonic anhydrase inhibitors for the treatment of epilepsy and obesity. In: Claudiu T. Supuran, Alessio Nocentini. Carbonic Anhydrases Biochemistry and Pharmacology of an Evergreen Pharmaceutical Target, pp. 311-329 Elsevier. DOI  

  Angeli A.; Ferraroni M.; Nocentini A.; Selleri S.; Gratteri P.; Supuran C.T.; Carta F. (2019). Polypharmacology of epacadostat: A potent and selective inhibitor of the tumor associated carbonic anhydrases IX and XII. CHEMICAL COMMUNICATIONS, vol. 55, pp. 5720-5723, ISSN:1359-7345 DOI   Accesso ONLINE all'editore

  Supuran C.T.; Altamimi A.S.A.; Carta F. (2019). Carbonic anhydrase inhibition and the management of glaucoma: a literature and patent review 2013-2019. EXPERT OPINION ON THERAPEUTIC PATENTS, vol. 29, pp. 781-792, ISSN:1354-3776 DOI   Accesso ONLINE all'editore

  Aspatwar A.; Kairys V.; Rala S.; Parikka M.; Bozdag M.; Carta F.; Supuran C.T.; Parkkila S. (2019). Mycobacterium tuberculosisβ-Carbonic Anhydrases: Novel Targets for Developing Antituberculosis Drugs. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, vol. 20, pp. 5153-5169, ISSN:1422-0067 DOI  

  Arias-Hidalgo, Mariela; Yuan, Qinggong; Carta, Fabrizio; Supuran, Claudiu T.; Gros, Gerolf; Endeward, Volker (2018). CO2Permeability of Rat Hepatocytes and Relation of CO2Permeability to CO2Production. CELLULAR PHYSIOLOGY AND BIOCHEMISTRY, vol. 46, pp. 1198-1208, ISSN:1015-8987 DOI   Accesso ONLINE all'editore

  Angeli A.; Trallori E.; Carta F.; Di Cesare Mannelli L.; Ghelardini C.; Supuran C.T. (2018). Heterocoumarins Are Selective Carbonic Anhydrase IX and XII Inhibitors with Cytotoxic Effects against Cancer Cells Lines. ACS MEDICINAL CHEMISTRY LETTERS, vol. 9, pp. 947-951, ISSN:1948-5875 DOI  

  Akgul, Ozlem; Di Cesare Mannelli, Lorenzo; Vullo, Daniela; Angeli, Andrea; Ghelardini, Carla; Bartolucci, Gianluca; Altamimi, Abdulmalik Saleh Alfawaz; Scozzafava, Andrea; Supuran, Claudiu T; Carta, Fabrizio (2018). Discovery of Novel Nonsteroidal Anti-Inflammatory Drugs and Carbonic Anhydrase Inhibitors Hybrids (NSAIDs-CAIs) for the Management of Rheumatoid Arthritis. JOURNAL OF MEDICINAL CHEMISTRY, pp. 1-60, ISSN:0022-2623 DOI  

  Bua, Silvia; Bozdag, Murat; Del Prete, Sonia; Carta, Fabrizio; Donald, William A; Capasso, Clemente; Supuran, Claudiu T (2018). Mono- and di-thiocarbamate inhibition studies of the δ-carbonic anhydrase TweCAδ from the marine diatom Thalassiosira weissflogii. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 33, pp. 707-713, ISSN:1475-6366 DOI  

  Nocentini, Alessio; Carta, Fabrizio; Tanc, Muhammet; Selleri, Silvia; Supuran, Claudiu T.; Bazzicalupi, Carla*; Gratteri, Paola (2018). Deciphering the Mechanism of Human Carbonic Anhydrases Inhibition with Sulfocoumarins: Computational and Experimental Studies. CHEMISTRY-A EUROPEAN JOURNAL, vol. 24, pp. 7840-7844, ISSN:0947-6539 DOI   Accesso ONLINE all'editore

  Supuran, Claudiu T.; Alterio, Vincenzo; Di Fiore, Anna; D' Ambrosio, Katia; Carta, Fabrizio; Monti, Simona Maria; De Simone, Giuseppina* (2018). Inhibition of carbonic anhydrase IX targets primary tumors, metastases, and cancer stem cells: Three for the price of one. MEDICINAL RESEARCH REVIEWS, pp. 1-38, ISSN:0198-6325 DOI   Accesso ONLINE all'editore

  Bua, Silvia; Berrino, Emanuela; Del Prete, Sonia; Murthy, Vallabhaneni S; Vijayakumar, Vijayaparthasarathi; Tamboli, Yasinalli; Capasso, Clemente; Cerbai, Elisabetta; Mugelli, Alessandro; Carta, Fabrizio; Supuran, Claudiu T (2018). Synthesis of novel benzenesulfamide derivatives with inhibitory activity against human cytosolic carbonic anhydrase I and II and Vibrio cholerae α- and β-class enzymes. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 33, pp. 1125-1136, ISSN:1475-6366 DOI  

  Provensi, G ; Schmidt, SD; Rani, B ; Costa, A ; Carta, F ; de Carvalho Myskiw, J.; Passani, MB ; Izquierdo, I ; Supuran, CT; Blandina P (2018). BRAIN CARBONIC ANHYDRASES INHIBITION IMPAIRS FEAR MEMORY EXTINCTION IN RATS. BASIC & CLINICAL PHARMACOLOGY & TOXICOLOGY, vol. 123, pp. 61-61, ISSN:1742-7835

  Logsdon, Derek P.; Shah, Fenil; Carta, Fabrizio; Supuran, Claudiu T.; Kamocka, Malgorzata; Jacobsen, Max H.; Sandusky, George E.; Kelley, Mark R.; Fishel, Melissa L. (2018). Blocking HIF signaling via novel inhibitors of CA9 and APE1/Ref-1 dramatically affects pancreatic cancer cell survival. SCIENTIFIC REPORTS, vol. 8, pp. 13759-13773, ISSN:2045-2322 DOI   Accesso ONLINE all'editore

  Angeli, Andrea; Trallori, Elena; Carta, Fabrizio; Di Cesare Mannelli, Lorenzo; Ghelardini, Carla; Supuran, Claudiu T.* (2018). Heterocoumarins Are Selective Carbonic Anhydrase IX and XII Inhibitors with Cytotoxic Effects against Cancer Cells Lines. ACS MEDICINAL CHEMISTRY LETTERS, vol. 9, pp. 947-951, ISSN:1948-5875 DOI   Accesso ONLINE all'editore

  Angeli, Andrea; Di Cesare Mannelli, Lorenzo; Trallori, Elena; Peat, Thomas S.; Ghelardini, Carla; Carta, Fabrizio; Supuran, Claudiu T.* (2018). Design, Synthesis, and X-ray of Selenides as New Class of Agents for Prevention of Diabetic Cerebrovascular Pathology. ACS MEDICINAL CHEMISTRY LETTERS, vol. 9, pp. 462-467, ISSN:1948-5875 DOI   Accesso ONLINE all'editore

  Aspatwar A.; Winum J.-Y.; Carta F.; Supuran C.T.; Hammaren M.; Parikka M.; Parkkila S. (2018). Carbonic anhydrase inhibitors as novel drugs against mycobacterial β-carbonic anhydrases: An update on in vitro and in vivo studies. MOLECULES, vol. 23, pp. 2911-2925, ISSN:1420-3049 DOI   Accesso ONLINE all'editore

  Mboge M.Y.; Chen Z.; Wolff A.; Mathias J.V.; Tu C.; Brown K.D.; Bozdag M.; Carta F.; Supuran C.T.; McKenna R.; Frost S.C. (2018). Selective inhibition of carbonic anhydrase IX over carbonic anhydrase XII in breast cancer cells using benzene sulfonamides: Disconnect between activity and growth inhibition. PLOS ONE, vol. 13, pp. e0207417--, ISSN:1932-6203 DOI  

  Carta F. (2018). Preface. CURRENT ENZYME INHIBITION, vol. 14, pp. 2-2, ISSN:1573-4080 Accesso ONLINE all'editore

  Nocentini, Alessio; Ceruso, Mariangela; Bua, Silvia; Lomelino, Carrie L.; Andring, Jacob T.; McKenna, Robert; Lanzi, Cecilia; Sgambellone, Silvia; Pecori, Riccardo; Matucci, Rosanna; Filippi, Luca; Gratteri, Paola; Carta, Fabrizio; Masini, Emanuela; Selleri, Silvia*; Supuran, Claudiu T. (2018). Discovery of β-Adrenergic Receptors Blocker-Carbonic Anhydrase Inhibitor Hybrids for Multitargeted Antiglaucoma Therapy. JOURNAL OF MEDICINAL CHEMISTRY, vol. 61, pp. 5380-5394, ISSN:0022-2623 DOI   Accesso ONLINE all'editore

  Bozdag M.; Carta F.; Angeli A.; Osman S.M.; Alasmary F.A.S.; AlOthman Z.; Supuran C.T. (2018). Synthesis of N′-phenyl-N-hydroxyureas and investigation of their inhibitory activities on human carbonic anhydrases. BIOORGANIC CHEMISTRY, vol. 78, pp. 1-6, ISSN:0045-2068 DOI   Accesso ONLINE all'editore

  Bozdag, Murat; Carta, Fabrizio; Ceruso, Mariangela; Ferraroni, Marta; McDonald, Paul C.; Dedhar, Shoukat; Supuran, Claudiu T.* (2018). Discovery of 4-Hydroxy-3-(3-(phenylureido)benzenesulfonamides as SLC-0111 Analogues for the Treatment of Hypoxic Tumors Overexpressing Carbonic Anhydrase IX. JOURNAL OF MEDICINAL CHEMISTRY, vol. 61, pp. 6328-6338, ISSN:0022-2623 DOI   Accesso ONLINE all'editore

  Menicatti, Marta; Pallecchi, Marco; Bua, Silvia; Vullo, Daniela; Di Cesare Mannelli, Lorenzo; Ghelardini, Carla; Carta, Fabrizio; Supuran, Claudiu T.; Bartolucci, Gianluca* (2018). Resolution of co-eluting isomers of anti-inflammatory drugs conjugated to carbonic anhydrase inhibitors from plasma in liquid chromatography by energy-resolved tandem mass spectrometry. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 33, pp. 671-679, ISSN:1475-6366 DOI  

  Vullo, Daniela; Del Prete, Sonia; Nocentini, Alessio; Osman, Sameh M.; Alothman, Zeid; Capasso, Clemente; Bozdag, Murat; Carta, Fabrizio; Gratteri, Paola; Supuran, Claudiu T. (2017). Dithiocarbamates effectively inhibit the β-carbonic anhydrase from the dandruff-producing fungus Malassezia globosa. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 25, pp. 1260-1265, ISSN:0968-0896 DOI   Accesso ONLINE all'editore

  Bozdag, Murat; Alafeefy, Ahmed Mahmoud; Altamimi, Abdul Malik; Vullo, Daniela; Carta, Fabrizio; Supuran, Claudiu T. (2017). Coumarins and other fused bicyclic heterocycles with selective tumor-associated carbonic anhydrase isoforms inhibitory activity. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 25, pp. 677-683, ISSN:0968-0896 DOI   Accesso ONLINE all'editore

  Bua, Silvia; Di Cesare Mannelli, Lorenzo; Vullo, Daniela; Ghelardini, Carla; Bartolucci, Gianluca; Scozzafava, Andrea; Supuran, Claudiu T; Carta, Fabrizio (2017). Design and Synthesis of Novel Nonsteroidal Anti-Inflammatory Drugs and Carbonic Anhydrase Inhibitors Hybrids (NSAIDs-CAIs) for the Treatment of Rheumatoid Arthritis. JOURNAL OF MEDICINAL CHEMISTRY, vol. 60, pp. 1159-1170, ISSN:0022-2623 DOI   Accesso ONLINE all'editore

  Bertol, Elisabetta; Vaiano, Fabio; Mari, Francesco; Di Milia, Maria Grazia; Bua, Silvia; Supuran, Claudiu Trandafir; Carta, Fabrizio (2017). Advances in New Psychoactive Substances Identification: The U.R.I.To.N Consortium. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 32, pp. 841-849, ISSN:1475-6366 DOI  

  Nocentini, Alessio; Vullo, Daniela; Del Prete, Sonia; Osman, Sameh M.; Alasmary, Fatmah A. S.; Alothman, Zeid; Capasso, Clemente; Carta, Fabrizio; Gratteri, Paola; Supuran, Claudiu T. (2017). Inhibition of the β-carbonic anhydrase from the dandruff-producing fungus Malassezia globosa with monothiocarbamates. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 32, pp. 1064-1070, ISSN:1475-6366 DOI   Accesso ONLINE all'editore

  Angeli, Andrea; Abbas, Ghulam; Del Prete, Sonia; Carta, Fabrizio; Capasso, Clemente; Supuran, Claudiu T. (2017). Acyl selenoureido benzensulfonamides show potent inhibitory activity against carbonic anhydrases from the pathogenic bacterium Vibrio cholerae. BIOORGANIC CHEMISTRY, vol. 75, pp. 170-172, ISSN:0045-2068 DOI   Accesso ONLINE all'editore

  Andreucci, Elena; Peppicelli, Silvia; Carta, Fabrizio; Brisotto, Giulia; Biscontin, Eva; Ruzzolini, Jessica; Bianchini, Francesca; Biagioni, Alessio; Supuran, Claudiu T.; Calorini, Lido (2017). Carbonic anhydrase IX inhibition affects viability of cancer cells adapted to extracellular acidosis. JOURNAL OF MOLECULAR MEDICINE, vol. 95, pp. 1341-1353, ISSN:0946-2716 DOI   Accesso ONLINE all'editore

  Bozdag, Murat; Alafeefy, Ahmed Mahmoud; Altamimi, Abdul Malik; Carta, Fabrizio; Supuran, Claudiu T.*; Vullo, Daniela (2017). Synthesis of new 3-(2-mercapto-4-oxo-4H-quinazolin-3-yl)-benzenesulfonamides with strong inhibition properties against the tumor associated carbonic anhydrases IX and XII. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 25, pp. 2782-2788, ISSN:0968-0896 DOI   Accesso ONLINE all'editore

  Carta, Fabrizio; Vullo, Daniela; Osman, Sameh M.; AlOthman, Zeid; Supuran, Claudiu T. (2017). Synthesis and carbonic anhydrase inhibition of a series of SLC-0111 analogs. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 25, pp. 2569-2576, ISSN:0968-0896 DOI   Accesso ONLINE all'editore

  Carta, Fabrizio*; Birkmann, Alexander; Pfaff, Tamara; Buschmann, Helmut; Schwab, Wilfried; Zimmermann, Holger; Maresca, Alfonso; Supuran, Claudiu T. (2017). Lead Development of Thiazolylsulfonamides with Carbonic Anhydrase Inhibitory Action. JOURNAL OF MEDICINAL CHEMISTRY, vol. 60, pp. 3154-3164, ISSN:0022-2623 DOI   Accesso ONLINE all'editore

  Angeli, Andrea; Carta, Fabrizio; Bartolucci, Gian Luca; Supuran, Claudiu T.* (2017). Synthesis of novel acyl selenoureido benzensulfonamides as carbonic anhydrase I, II, VII and IX inhibitors. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 25, pp. 3567-3573, ISSN:0968-0896 DOI   Accesso ONLINE all'editore

  Abdoli M.; Angeli A.; Bozdag M.; Carta F.; Kakanejadifard A.; Saeidian H.; Supuran C.T. (2017). Synthesis and carbonic anhydrase I, II, VII, and IX inhibition studies with a series of benzo[d]thiazole-5- and 6-sulfonamides. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 32, pp. 1071-1078, ISSN:1475-6366 DOI  

  Lucas Canto de Souza, Gustavo Provensi, Daniela Vullo, Fabrizio Carta, Andrea Scozzafava, Alessia Costa, Scheila D. Schmidt; Maria Beatrice Passani, Claudiu T. Supuran, Patrizio Blandina (2017). Carbonic anhydrase activation enhances object recognition memory in mice through phosphorylation of the extracellular signal-regulated kinase in the cortex and the hippocampus.. NEUROPHARMACOLOGY, vol. 118, pp. 148-156, ISSN:1873-7064 DOI   Accesso ONLINE all'editore

  Ivanova J.; Carta F.; Vullo D.; Leitans J.; Kazaks A.; Tars K.; Zalubovskis R.; Supuran C.T. (2017). N-Substituted and ring opened saccharin derivatives selectively inhibit transmembrane, tumor-associated carbonic anhydrases IX and XII. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 25, pp. 3583-3589, ISSN:0968-0896 DOI  

  Kusuzaki K.; Matsubara T.; Murata H.; Logozzi M.; Iessi E.; Di Raimo R.; Carta F.; Supuran C.T.; Fais S. (2017). Natural extracellular nanovesicles and photodynamic molecules: is there a future for drug delivery?. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 32, pp. 908-916, ISSN:1475-6366 DOI  

  Mboge M.Y.; Mahon B.P.; Lamas N.; Socorro L.; Carta F.; Supuran C.T.; Frost S.C.; McKenna R. (2017). Structure activity study of carbonic anhydrase IX: Selective inhibition with ureido-substituted benzenesulfonamides. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 132, pp. 184-191, ISSN:0223-5234 DOI  

  Aspatwar A.; Hammaren M.; Koskinen S.; Luukinen B.; Barker H.; Carta F.; Supuran C.T.; Parikka M.; Parkkila S. (2017). β-CA-specific inhibitor dithiocarbamate Fc14–584B: a novel antimycobacterial agent with potential to treat drug-resistant tuberculosis. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 32, pp. 832-840, ISSN:1475-6366 DOI  

  Meehan J.; Ward C.; Turnbull A.; Bukowski-Wills J.; Finch A.J.; Jarman E.J.; Xintaropoulou C.; Martinez-Perez C.; Gray M.; Pearson M.; Mullen P.; Supuran C.T.; Carta F.; Harrison D.J.; Kunkler I.H.; Langdon S.P. (2017). Inhibition of pH regulation as a therapeutic strategy in hypoxic human breast cancer cells. ONCOTARGET, vol. 8, pp. 42857-42875, ISSN:1949-2553 DOI  

  Bragagni M.; Carta F.; Osman S.M.; AlOthman Z.; Supuran C.T. (2017). Synthesis of an acridine orange sulfonamide derivative with potent carbonic anhydrase IX inhibitory action. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 32, pp. 701-706, ISSN:1475-6366 DOI  

  Angeli, Andrea; Tanini, Damiano; Peat, Thomas S. ; Di Cesare Mannelli,Lorenzo; Bartolucci, Gian Luca; Capperucci, Antonella; Ghelardini, Carla; Supuran, Claudiu T.; and Carta, Fabrizio (2017). Discovery of New Selenoureido Analogues of 4-(4-Fluorophenylureido)benzenesulfonamide as Carbonic Anhydrase Inhibitors. ACS MEDICINAL CHEMISTRY LETTERS, vol. 8, pp. 963-968, ISSN:1948-5875 DOI   Accesso ONLINE all'editore

  Berrino, Emanuela; Bua, Silvia; Mori, Mattia; Botta, Maurizio; Murthy, Vallabhaneni S.; Vijayakumar, Vijayaparthasarathi; Tamboli, Yasinalli; Bartolucci, Gianluca; Mugelli, Alessandro; Cerbai, Elisabetta; Supuran, Claudiu T.; Carta, Fabrizio (2017). Novel sulfamide-containing compounds as selective carbonic anhydrase i inhibitors. MOLECULES, vol. 22, pp. 1049-1065, ISSN:1420-3049 DOI   Accesso ONLINE all'editore

  Carta, Fabrizio; Ferraroni, Marta; Scozzafava, Andrea; Supuran, Claudiu T (2016). Fluorescent sulfonamide carbonic anhydrase inhibitors incorporating 1,2,3-triazole moieties: Kinetic and X-ray crystallographic studies. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 24, pp. 104-12-112, ISSN:0968-0896 DOI  

  Angeli, A; Peat, T.S.; Bartolucci, G.; Nocentini, A.; Supuran, C.T.; Carta, F. (2016). Intramolecular oxidative deselenization of acylselenoureas: a facile synthesis of benzoxazole amides and carbonic anhydrase inhibitors. ORGANIC & BIOMOLECULAR CHEMISTRY, vol. 14, pp. 11353-11356, ISSN:1477-0520 DOI   Accesso ONLINE all'editore

  Vullo, Daniela; Durante, Mariaconcetta; Di Leva, Francesco Saverio; Cosconati, Sandro; Masini, Emanuela; Scozzafava, Andrea; Novellino, Ettore; Supuran, Claudiu T.; Carta, Fabrizio (2016). Monothiocarbamates Strongly Inhibit Carbonic Anhydrases in Vitro and Possess Intraocular Pressure Lowering Activity in an Animal Model of Glaucoma. JOURNAL OF MEDICINAL CHEMISTRY, vol. 59, pp. 5857-5867, ISSN:0022-2623 DOI   Accesso ONLINE all'editore

  Ferraroni, Marta; Carta, Fabrizio; Scozzafava, Andrea; Supuran, Claudiu T. (2016). Thioxocoumarins Show an Alternative Carbonic Anhydrase Inhibition Mechanism Compared to Coumarins. JOURNAL OF MEDICINAL CHEMISTRY, vol. 59, pp. 462-473, ISSN:0022-2623 DOI   Accesso ONLINE all'editore

  Cornelio, Benedetta; Laronze Cochard, Marie; Ceruso, Mariangela; Ferraroni, Marta; Rance, Graham A.; Carta, Fabrizio; Khlobystov, Andrei N.; Fontana, Antonella; Supuran, CLAUDIU TRANDAFIR; Sapi, Janos (2016). 4-Arylbenzenesulfonamides as Human Carbonic Anhydrase Inhibitors (hCAIs): Synthesis by Pd Nanocatalyst-Mediated Suzuki-Miyaura Reaction, Enzyme Inhibition, and X-ray Crystallographic Studies. JOURNAL OF MEDICINAL CHEMISTRY, vol. 59, pp. 721-732, ISSN:0022-2623 DOI   Accesso ONLINE all'editore

  Margheri, F; Ceruso, M; Carta, F; Laurenzana, A; Maggi, L; Lazzeri, S; Simonini, G; Annunziato, F; Del Rosso, M; Supuran, CT; Cimaz, R (2016). Overexpression of the transmembrane carbonic anhydrase isoforms IX and XII in the inflamed synovium. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, pp. 0-0, ISSN:1475-6366 DOI  

  Nocentini, Alessio; Ceruso, Mariangela; Carta, Fabrizio; Supuran, Claudiu T. (2016). 7-Aryl-triazolyl-substituted sulfocoumarins are potent, selective inhibitors of the tumor-associated carbonic anhydrase IX and XII. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 31, pp. 1226-1233, ISSN:1475-6366 DOI  

  Lomelino, Carrie L.; Mahon, Brian P.; Mckenna, Robert; Carta, Fabrizio; Supuran, Claudiu T. (2016). Kinetic and X-ray crystallographic investigations on carbonic anhydrase isoforms I, II, IX and XII of a thioureido analog of SLC-0111. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 24, pp. 976-981, ISSN:0968-0896 DOI   Accesso ONLINE all'editore

  Di Fiore, Anna; De Simone, Giuseppina; Alterio, Vincenzo; Riccio, Vincenzo; Winum, Jean-Yves; Carta, Fabrizio; Supuran, Claudiu T. (2016). The anticonvulsant sulfamide JNJ-26990990 and its: S, S -dioxide analog strongly inhibit carbonic anhydrases: Solution and X-ray crystallographic studies. ORGANIC & BIOMOLECULAR CHEMISTRY, vol. 14, pp. 4853-4858, ISSN:1477-0520 DOI   Accesso ONLINE all'editore

  van Kuijk, Simon J.A; Parvathaneni, Nanda Kumar; Niemans, Raymon; van Gisbergen, Marike W.; Carta, Fabrizio; Vullo, Daniela; Pastorekova, Silvia; Yaromina, Ala; Supuran, Claudiu T.; Dubois, Ludwig J.; Winum, Jean-Yves; Lambin, Philippe (2016). New approach of delivering cytotoxic drugs towards CAIX expressing cells: A concept of dual-target drugs. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 127, pp. 691-702, ISSN:0223-5234 DOI   Accesso ONLINE all'editore

  Karioti, Anastasia; Carta, Fabrizio; Supuran, Claudiu T. (2016). Phenols and polyphenols as Carbonic anhydrase inhibitors. MOLECULES, vol. 21, pp. 1649-1676, ISSN:1420-3049 DOI   Accesso ONLINE all'editore

  Arias-Hidalgo, Mariela; Hegermann, Jan; Tsiavaliaris, Georgios; Carta, Fabrizio; Supuran, Claudiu T.; Gros, Gerolf; Endeward, Volker (2016). CO2 and HCO3- Permeability of the Rat Liver Mitochondrial Membrane. CELLULAR PHYSIOLOGY AND BIOCHEMISTRY, vol. 39, pp. 2014-2024, ISSN:1015-8987 DOI   Accesso ONLINE all'editore

  Bozdag, Murat; Carta, Fabrizio; Vullo, Daniela*; Isik, Semra; AlOthman, Zeid; Osman, Sameh M.; Scozzafava, Andrea; Supuran, Claudiu T. (2016). Dithiocarbamates with potent inhibitory activity against the Saccharomyces cerevisiae β-carbonic anhydrase. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 31, pp. 132-136, ISSN:1475-6366 DOI  

  Nocentini, Alessio; Ferraroni, Marta; Carta, Fabrizio; Ceruso, Mariangela; Gratteri, Paola; Lanzi, Cecilia; Masini, Emanuela; Supuran, Claudiu T (2016). Benzenesulfonamides Incorporating Flexible Triazole Moieties Are Highly Effective Carbonic Anhydrase Inhibitors: Synthesis and Kinetic, Crystallographic, Computational, and Intraocular Pressure Lowering Investigations. JOURNAL OF MEDICINAL CHEMISTRY, vol. 59, pp. 10692-10704, ISSN:0022-2623 DOI   Accesso ONLINE all'editore

  Vullo, Daniela; Supuran, Claudiu T.; Scozzafava, Andrea; De Simone, Giuseppina; Monti, Simona Maria; Alterio, Vincenzo; Carta, Fabrizio (2016). Kinetic and X-ray crystallographic investigations of substituted 2-thio-6-oxo-1,6-dihydropyrimidine–benzenesulfonamides acting as carbonic anhydrase inhibitors. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 24, pp. 3643-3648, ISSN:0968-0896 DOI   Accesso ONLINE all'editore

  Federici, Cristina; Lugini, Luana; Marino, Maria Lucia; Carta, Fabrizio; Iessi, Elisabetta; Azzarito, Tommaso; Supuran, Claudiu T.; Fais, Stefano (2016). Lansoprazole and carbonic anhydrase IX inhibitors sinergize against human melanoma cells. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 31, pp. 119-125, ISSN:1475-6366 DOI  

  Alafeefy, Ahmed M; Carta, Fabrizio; Ceruso, Mariangela; Al-Tamimi, Abdul-Malek S; Al-Kahtani, Abdulla A; Supuran, Claudiu T (2016). Development of 3-(4-aminosulphonyl)-phenyl-2-mercapto-3H-quinazolin-4-ones as inhibitors of carbonic anhydrase isoforms involved in tumorigenesis and glaucoma. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 24, pp. 1402-1407, ISSN:0968-0896 DOI  

  Scozzafava, Andrea; Supuran, Claudiu T; Carta, Fabrizio (2016). Polyamines and α-carbonic anhydrases. MOLECULES, vol. 21, pp. 1726-1735, ISSN:1420-3049 DOI   Accesso ONLINE all'editore

  Karioti, Anastasia; Carta, Fabrizio; Supuran, Claudiu (2016). An Update on Natural Products with Carbonic Anhydrase Inhibitory Activity. CURRENT PHARMACEUTICAL DESIGN, vol. 22, pp. 1570-1591, ISSN:1381-6128 DOI  

  Bozdag, Murat; Alafeefy, Ahmed M.; Carta, Fabrizio; Ceruso, Mariangela; Al-Tamimi, Abdul-Malek S.; Al-Kahtani, Abdulla A.; Alasmary, Fatmah A.S.; Supuran, Claudiu T (2016). Synthesis 4-[2-(2-mercapto-4-oxo-4H-quinazolin-3-yl)-ethyl]-benzenesulfonamides with subnanomolar carbonic anhydrase II and XII inhibitory properties. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 24, pp. 4100-4107, ISSN:0968-0896 DOI   Accesso ONLINE all'editore

  Logsdon, Derek P.; Grimard, Michelle; Luo, Meihua; Shahda, Safi; Jiang, Yanlin; Tong, Yan; Yu, Zhangsheng; Zyromski, Nicholas; Schipani, Ernestina; Carta, Fabrizio; Supuran, Claudiu T.; Korc, Murray; Ivan, Mircea; Kelley, Mark R.; Fishel, Melissa L. (2016). Regulation of HIF1a under hypoxia by APE1/Ref-1 impacts CA9 expression: Dual targeting in patient-derived 3D pancreatic cancer models. MOLECULAR CANCER THERAPEUTICS, vol. 15, pp. 2722-2732, ISSN:1535-7163 DOI   Accesso ONLINE all'editore

  Alafeefy, Ahmed M.; Ahmad, Rehan; Abdulla, Maha; Eldehna, Wagdy M.; Al-Tamimi, Abdul-Malek S.; Abdel-Aziz, Hatem A.; Al-Obaid, Omar; Carta, Fabrizio; Al-Kahtani, Abdulla A.; Supuran, Claudiu T. (2016). Development of certain new 2-substituted-quinazolin-4-ylaminobenzenesulfonamide as potential antitumor agents. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 109, pp. 247-253, ISSN:0223-5234 DOI   Accesso ONLINE all'editore

  M. Tanc;F. Carta;A. Scozzafava;C. T. Supuran (2015). 6-Substituted 1,2-benzoxathiine-2,2-dioxides are isoform-selective inhibitors of human carbonic anhydrases IX, XII and VA.. ORGANIC & BIOMOLECULAR CHEMISTRY, vol. 13, pp. 77-80, ISSN:1477-0520 DOI   Accesso ONLINE all'editore

  Karioti, Anastasia; Ceruso, Mariangela; Carta, Fabrizio; Bilia, Anna-Rita; Supuran, Claudiu T (2015). New natural product carbonic anhydrase inhibitors incorporating phenol moieties. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 23, pp. 7219-25-7225, ISSN:0968-0896 DOI  

  Perut, Francesca; Carta, Fabrizio; Bonuccelli, Gloria; Grisendi, Giulia; Di Pompo, Gemma; Avnet, Sofia; Sbrana, Francesca Vittoria; Hosogi, Shigekuni; Dominici, Massimo; Kusuzaki, Katsuyuki; Supuran, Claudiu T; Baldini, Nicola (2015). Carbonic anhydrase IX inhibition is an effective strategy for osteosarcoma treatment. EXPERT OPINION ON THERAPEUTIC TARGETS, pp. 1-13, ISSN:1472-8222 DOI  

  Carta, Fabrizio; Osman, Sameh M.; Vullo, Daniela; Alothman, Zeid; Supuran, Claudiu T. (2015). Dendrimers incorporating benzenesulfonamide moieties strongly inhibit carbonic anhydrase isoforms I-XIV. ORGANIC & BIOMOLECULAR CHEMISTRY, vol. 13, pp. 6453-6457, ISSN:1477-0520 DOI   Accesso ONLINE all'editore

  Tanc, Muhammet; Carta, Fabrizio; Scozzafava, Andrea; Supuran, Claudiu T. (2015). α-carbonic anhydrases possess thioesterase activity. ACS MEDICINAL CHEMISTRY LETTERS, vol. 6, pp. 292-295, ISSN:1948-5875 DOI   Accesso ONLINE all'editore

  Carta, Fabrizio; Di Cesare Mannelli, Lorenzo; Pinard, Melissa; Ghelardini, Carla; Scozzafava, Andrea; Mckenna, Robert; Supuran, Claudiu T. (2015). A class of sulfonamide carbonic anhydrase inhibitors with neuropathic pain modulating effects. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 23, pp. 1828-1840, ISSN:0968-0896 DOI   Accesso ONLINE all'editore

  Ceruso, Mariangela; Carta, Fabrizio; Osman, Sameh M.; Alothman, Zeid; Monti, Simona Maria; Supuran, Claudiu T. (2015). Inhibition studies of bacterial, fungal and protozoan β-class carbonic anhydrases with Schiff bases incorporating sulfonamide moieties. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 23, pp. 4181-4187, ISSN:0968-0896 DOI   Accesso ONLINE all'editore

  Bragagni, Marco; Bozdag, Murat; Carta, Fabrizio; Scozzafava, Andrea; Lanzi, Cecilia; Masini, Emanuela; Mura, Paola; Supuran, Claudiu T. (2015). Cyclodextrin complexation highly enhances efficacy of arylsulfonylureido benzenesulfonamide carbonic anhydrase inhibitors as a topical antiglaucoma agents. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 23, pp. 6223-6227, ISSN:1464-3391 DOI   Accesso ONLINE all'editore

  Di Cesare Mannelli, Lorenzo; Micheli, Laura; Carta, Fabrizio; Cozzi, Andrea; Ghelardini, Carla; Supuran, Claudiu T (2015). Carbonic anhydrase inhibition for the management of cerebral ischemia: in vivo evaluation of sulfonamide and coumarin inhibitors. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, pp. 1-6, ISSN:1475-6366 DOI  

  Carta, Fabrizio; Osman, Sameh M.; Vullo, Daniela; Gullotto, Antonella; Winum, Jean-Yves; Alothman, Zeid; Masini, Emanuela; Supuran, Claudiu T. (2015). Poly(amidoamine) dendrimers with carbonic anhydrase inhibitory activity and antiglaucoma action. JOURNAL OF MEDICINAL CHEMISTRY, vol. 58, pp. 4039-4045, ISSN:0022-2623 DOI   Accesso ONLINE all'editore

  Bozdag, Murat; Carta, Fabrizio; Vullo, Daniela; Akdemir, Atilla; Isik, Semra; Lanzi, Cecilia; Scozzafava, Andrea; Masini, Emanuela; Supuran, Claudiu T. (2015). Synthesis of a new series of dithiocarbamates with effective human carbonic anhydrase inhibitory activity and antiglaucoma action. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 23, pp. 2368-2376, ISSN:0968-0896 DOI   Accesso ONLINE all'editore

  Nocentini, Alessio; Carta, Fabrizio; Ceruso, Mariangela; Bartolucci, Gianluca; Supuran, Claudiu T. (2015). Click-tailed coumarins with potent and selective inhibitory action against the tumor-associated carbonic anhydrases IX and XII. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 23, pp. 6955-6966, ISSN:0968-0896 DOI   Accesso ONLINE all'editore

  Carta, Fabrizio; Osman, Sameh M.; Vullo, Daniela; Alothman, Zeid; Del Prete, Sonia; Capasso, Clemente; Supuran, Claudiu T. (2015). Poly(amidoamine) dendrimers show carbonic anhydrase inhibitory activity against α-, β-, γ- and η-class enzymes. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 23, pp. 6794-6798, ISSN:0968-0896 DOI   Accesso ONLINE all'editore

  Trabocchi, Andrea; Pala, N.; Krimmelbein, I.; Menchi, Gloria; Guarna, Antonio; Sechi, M.; Dreker, T.; Scozzafava, Andrea; Supuran, CLAUDIU TRANDAFIR; Carta, Fabrizio (2015). Peptidomimetics as protein arginine deiminase 4 (PAD4) inhibitors.. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 30, pp. 466-471, ISSN:1475-6366 DOI   Accesso ONLINE all'editore

  José, O.; Torres-Rodríguez, P.; Forero-Quintero, L.S.; Chávez, J.C.; De La Vega-Beltrán, J.L.; Carta, F.; Supuran, C.T.; Deitmer, J.W.; Treviño, C.L.* (2015). Carbonic anhydrases and their functional differences in human and mouse sperm physiology. BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, vol. 468, pp. 713-718, ISSN:0006-291X DOI   Accesso ONLINE all'editore

  Alafeefy, Ahmed M.*; Abdel-Aziz, Hatem A.; Carta, F.; Supuran, Claudiu T.; Pathak, Shilendra K.; Prasad, Onkar; Sinha, Leena (2015). Exploring QSARs of some benzenesulfonamides incorporating cyanoacrylamide moieties as a carbonic anhydrase inhibitors (specifically against tumor-associated isoforms IX and XII). JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 30, pp. 519-523, ISSN:1475-6366 DOI  

  Vullo, Daniela*; Isik, Semra; Bozdag, Murat; Carta, Fabrizio; Supuran, Claudiu T. (2015). 7-Amino-3,4-dihydro-1H-quinolin-2-one, a compound similar to the substituted coumarins, inhibits α-carbonic anhydrases without hydrolysis of the lactam ring.. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 30, pp. 773-777, ISSN:1475-6366 DOI   Accesso ONLINE all'editore

  Fulvio Ratto; Ewa Witort; Francesca Tatini; Sonia Centi; Lorenza Lazzeri; Fabrizio Carta; Matteo Lulli; Daniela Vullo; Franco Fusi; Claudiu T. Supuran; Andrea Scozzafava; Sergio Capaccioli; Roberto Pini (2015). Plasmonic Particles that Hit Hypoxic Cells. ADVANCED FUNCTIONAL MATERIALS, vol. 25, pp. 316-323, ISSN:1616-3028 DOI  

  Grandane, Aiga; Tanc, Muhammet; Di Cesare Mannelli, Lorenzo; Carta, Fabrizio; Ghelardini, Carla; Žalubovskis, Raivis; Supuran, Claudiu T. (2015). 6-substituted sulfocoumarins are selective carbonic anhdydrase IX and XII Inhibitors with significant cytotoxicity against colorectal cancer cells. JOURNAL OF MEDICINAL CHEMISTRY, vol. 58, pp. 3975-3983, ISSN:0022-2623 DOI   Accesso ONLINE all'editore

  Bozdag, Murat; Alafeefy, Ahmed M.; Vullo, Daniela; Carta, Fabrizio; Dedeoglu, Nurcan; Al-Tamimi, Abdul-Malek S.; Al-Jaber, Nabila A.; Scozzafava, Andrea; Supuran, Claudiu T (2015). Benzenesulfonamides incorporating bulky aromatic/heterocyclic tails with potent carbonic anhydrase inhibitory activity. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 23, pp. 7751-7764, ISSN:0968-0896 DOI   Accesso ONLINE all'editore

  Sethi, Kalyan K; Verma, Saurabh M.; Tanç, Muhammet; Purper, Gaultier; Calafato, Gaetan; Carta, Fabrizio; Supuran, Claudiu T. (2014). Carbonic anhydrase inhibitors: Synthesis and inhibition of the human carbonic anhydrase isoforms I, II, IX and XII with benzene sulfonamides incorporating 4- and 3-nitrophthalimide moieties. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 22, pp. 1586-1595, ISSN:0968-0896 DOI  

  F. Carta;C. T. Supuran;A. Scozzafava (2014). Sulfonamides and their isosters as carbonic anhydrase inhibitors.. FUTURE MEDICINAL CHEMISTRY, vol. 6, pp. 1149-1165, ISSN:1756-8919 DOI   Accesso ONLINE all'editore

  Sarikaya, Busra; Ceruso, Mariangela; Carta, Fabrizio; Supuran, Claudiu T. (2014). Inhibition of carbonic anhydrase isoforms I, II, IX and XII with novel Schiff bases: Identification of selective inhibitors for the tumor-associated isoforms over the cytosolic ones. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 22, pp. 5883-5890, ISSN:0968-0896 DOI   Accesso ONLINE all'editore

  K. Chegaev;L. Lazzarato;Y. Tamboli;D. Boschi;M. Blangetti;A. Scozzafava;F. Carta;E. Masini;R. Fruttero;C. T. Supuran;A. Gasco (2014). Furazan and furoxan sulfonamides are strong α-carbonic anhydrase inhibitors and potential antiglaucoma agents.. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 22, pp. 3913-3921, ISSN:0968-0896 DOI   Accesso ONLINE all'editore

  M. Bozdag;M. Ferraroni;F. Carta;D. Vullo;L. Lucarini;E. Orlandini;A. Rossello;E. Nuti;A. Scozzafava;E. Masini;C. T. Supuran (2014). Structural insights on carbonic anhydrase inhibitory action, isoform selectivity, and potency of sulfonamides and coumarins incorporating arylsulfonylureido groups.. JOURNAL OF MEDICINAL CHEMISTRY, vol. 57, pp. 9152-9167, ISSN:0022-2623 DOI   Accesso ONLINE all'editore

  Carta, Fabrizio*; Scozzafava, Andrea (2014). Next-generation polyamine human carbonic anhydrase inhibitors. In: Claudiu T Supuran e Clemente Capasso. Targeting Carbonic Anhydrases, pp. 68-81 Future medicine, ISBN:978-1-909453-91-3. DOI   Accesso ONLINE all'editore

  Carta, Fabrizio*; Bozdag, Murat; Tanc, Muhammet; Supuran, Claudiu (2014). Next-generation dithiocarbamate carbonic anhydrase inhibitors. In: Claudiu T Supuran e Clemente Capasso (editors). Targeting Carbonic Anhydrases, pp. 114-130 Future Medicine Ltd., ISBN:978-190945391-3. DOI   Accesso ONLINE all'editore

  Pala, Nicolino; Micheletto, Laura; Sechi, Mario; Aggarwal, Mayank; Carta, Fabrizio; Mckenna, Robert; Supuran, Claudiu T. (2014). Carbonic anhydrase inhibition with benzenesulfonamides and tetrafluorobenzenesulfonamides obtained via click chemistry. ACS MEDICINAL CHEMISTRY LETTERS, vol. 5, pp. 927-930, ISSN:1948-5875 DOI   Accesso ONLINE all'editore

  M. Bozdag;M. Ferraroni;E. Nuti;D. Vullo;A. Rossello;F. Carta;A. Scozzafava;C. T. Supuran (2014). Combining the tail and the ring approaches for obtaining potent and isoform-selective carbonic anhydrase inhibitors: solution and X-ray crystallographic studies.. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 22, pp. 334-340, ISSN:0968-0896 DOI   Accesso ONLINE all'editore

  M. Bozdag;M. Pinard;F. Carta;E. Masini;A. Scozzafava;R. McKenna;C. T. Supuran (2014). A class of 4-Sulfamoylphenyl-ω-aminoalkyl ethers with effective carbonic anhydrase inhibitory action and antiglaucoma effects.. JOURNAL OF MEDICINAL CHEMISTRY, vol. 57, pp. 9673-9686, ISSN:0022-2623 DOI   Accesso ONLINE all'editore

  C. T. Supuran;F. Carta;A. Scozzafava (2013). Metalloenzyme inhibitors for the treatment of Gram-negative bacterial infections: a patent review (2009 - 2012).. EXPERT OPINION ON THERAPEUTIC PATENTS, pp. 777-788, ISSN:1354-3776 DOI   Accesso ONLINE all'editore

  CLAUDIU SUPURAN; ANDREA SCOZZAFAVA; EMANUELA MASINI; FABRIZIO CARTA; ERIK OLAI PETTERSEN; PETER EBBERSEN (2013). A CARBONIC ANHYDRASE INHIBITOR COMPRISING A DITHIOCARBAMATE. Numero: WO 2013/050426 A1 CLAUDIU SUPURAN, ANDREA SCOZZAFAVA, EMANUELA MASINI, FABRIZIO CARTA, ERIK OLAI PETTERSEN, PETER EBBERSEN

  F. Bellissima;F. Carta;A. Innocenti;A. Scozzafava;P. Baglioni;C. T. Supuran;D. Berti (2013). Structural modulation of the biological activity of gold nanoparticles functionalized with a carbonic anhydrase inhibitor.. THE EUROPEAN PHYSICAL JOURNAL. E, SOFT MATTER, vol. 36, pp. 48-57, ISSN:1292-8941 DOI   Accesso ONLINE all'editore

  M. Tanc;F. Carta;M. Bozdag;A. Scozzafava;C. T. Supuran (2013). 7-Substituted-sulfocoumarins are isoform-selective, potent carbonic anhydrase II inhibitors.. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 21, pp. 4502-4510, ISSN:0968-0896 DOI   Accesso ONLINE all'editore

  H. M. Said;C. Hagemann;F. Carta;A. Katzer;B. Polat;A. Staab;A. Scozzafava;J. Anacker;G. H. Vince;M. Flentje;C. T. Supuran (2013). Hypoxia induced CA9 inhibitory targeting by two different sulfonamide derivatives including acetazolamide in human glioblastoma.. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 21, pp. 3949-3957, ISSN:0968-0896 DOI   Accesso ONLINE all'editore

  Sethi, Kalyan K; Vullo, Daniella; Verma, Saurabh M.; Tanç, Muhammet; Carta, Fabrizio; Supuran, Claudiu T. (2013). Carbonic anhydrase inhibitors: Synthesis and inhibition of the human carbonic anhydrase isoforms I, II, VII, IX and XII with benzene sulfonamides incorporating 4,5,6,7-tetrabromophthalimide moiety. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 21, pp. 5973-5982, ISSN:0968-0896 DOI  

  Sethi, Kalyan K; Verma, Saurabh M.; Tanç, Muhammet; Carta, Fabrizio; Supuran, Claudiu T. (2013). Carbonic anhydrase inhibitors: Synthesis and inhibition of the cytosolic mammalian carbonic anhydrase isoforms I, II and VII with benzene sulfonamides incorporating 4,5,6,7-tetrachlorophthalimide moiety. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 21, pp. 5168-5174, ISSN:0968-0896 DOI  

  E. Masini;F. Carta;A. Scozzafava;C. T. Supuran (2013). Antiglaucoma carbonic anhydrase inhibitors: a patent review.. EXPERT OPINION ON THERAPEUTIC PATENTS, vol. 23, pp. 705-716, ISSN:1354-3776 DOI   Accesso ONLINE all'editore

  F. Carta;A. Akdemir;A. Scozzafava;E. Masini;C. T. Supuran (2013). Xanthates and Trithiocarbonates Strongly Inhibit Carbonic Anhydrases and Show Antiglaucoma Effects in Vivo.. JOURNAL OF MEDICINAL CHEMISTRY, pp. 4691-4700, ISSN:0022-2623 DOI   Accesso ONLINE all'editore

  F. Carta;D. Vullo;A. Maresca;A. Scozzafava;C. T. Supuran (2013). Mono-/dihydroxybenzoic acid esters and phenol pyridinium derivatives as inhibitors of the mammalian carbonic anhydrase isoforms I, II, VII, IX, XII and XIV.. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 6, pp. 1564-1569, ISSN:0968-0896 DOI   Accesso ONLINE all'editore

  Roberto Pini; Fulvio RATTO; Francesca TATINI; Franco Fusi; Sonia CENTI; Andrea Scozzafava; Claudiu Trandafir SUPURAN; Fabrizio Carta; Sergio Capaccioli; Ewa Janina WITORT (2013). Assembly comprising an absorber of near infrared (nir) light covalently linked to an inhibitor of carbonic anhydrase. Numero: EP2964272 CNR

  Tania Fiaschi;Elisa Giannoni;Maria Letizia Taddei;Paolo Cirri;Alberto Marini;Gianfranco Pintus;Cristina Nativi;Barbara Richichi;Andrea Scozzafava;Fabrizio Carta;Eugenio Torre;Claudiu T. Supuran;Paola Chiarugi (2013). Carbonic anhydrase IX from cancer-associated fibroblasts drives epithelial-mesenchymal transition in prostate carcinoma cells. CELL CYCLE, vol. 12, pp. 1791-1801, ISSN:1538-4101 DOI  

  Carta, Fabrizio; Supuran, Claudiu T (2013). Diuretics with carbonic anhydrase inhibitory action: A patent and literature review (2005-2013). EXPERT OPINION ON THERAPEUTIC PATENTS, vol. 23, pp. 681-691, ISSN:1354-3776 DOI  

  Biswas, Shyamasri; Carta, Fabrizio; Scozzafava, Andrea; McKenna, Robert*; Supuran, Claudiu T. (2013). Structural effect of phenyl ring compared to thiadiazole based adamantyl-sulfonamides on carbonic anhydrase inhibition. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 21, pp. 2314-2318, ISSN:0968-0896 DOI  

  Bozdag, Murat; Dreker, Tobias; Henry, Christophe; Tosco, Paolo; Vallaro, Maura; Fruttero, Roberta; Scozzafava, Andrea; Carta, Fabrizio*; Supuran, Claudiu T. (2013). Novel small molecule protein arginine deiminase 4 (PAD4) inhibitors. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 23, pp. 715-719, ISSN:0960-894X DOI  

  A. Scozzafava;C. T. Supuran;F. Carta (2013). Antiobesity carbonic anhydrase inhibitors: a literature and patent review.. EXPERT OPINION ON THERAPEUTIC PATENTS, vol. 23, pp. 725-735, ISSN:1354-3776 DOI   Accesso ONLINE all'editore

  L. Syrjänen;M. E. E;M. Hilvo;D. Vullo;F. Carta;C. T. Supuran;S. Parkkila (2013). Characterization, bioinformatic analysis and dithiocarbamate inhibition studies of two new α-carbonic anhydrases, CAH1 and CAH2, from the fruit fly Drosophila melanogaster.. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 21, pp. 1516-1521, ISSN:0968-0896 DOI   Accesso ONLINE all'editore

  F. Carta;A. Maresca;A. Scozzafava;C. T. Supuran (2012). 5- and 6-membered (thio)lactones are prodrug type carbonic anhydrase inhibitors.. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 22, pp. 267-270, ISSN:0960-894X DOI   Accesso ONLINE all'editore

  S. Parkkila;D. Vullo;A. Maresca;F. Carta;A. Scozzafava;C. T. Supuran (2012). Serendipitous fragment-based drug discovery: ketogenic diet metabolites and statins effectively inhibit several carbonic anhydrases.. CHEMICAL COMMUNICATIONS, vol. 48, pp. 3551-3553, ISSN:1364-548X DOI   Accesso ONLINE all'editore

  J. Winum;F. Carta;C. Ward;P. Mullen;D. Harrison;S. P. Langdon;A. Cecchi;A. Scozzafava;I. Kunkler;C. T. Supuran (2012). Ureido-substituted sulfamates show potent carbonic anhydrase IX inhibitory and antiproliferative activities against breast cancer cell lines.. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 22(14), pp. 4681-4685, ISSN:0960-894X DOI   Accesso ONLINE all'editore

  F. Carta;D. Vullo;A. Maresca;A. Scozzafava;C. T. Supuran (2012). New chemotypes acting as isozyme-selective carbonic anhydrase inhibitors with low affinity for the offtarget cytosolic isoform II.. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 22, pp. 2182-2185, ISSN:0960-894X DOI   Accesso ONLINE all'editore

  K. D'Ambrosio;F. Smaine;F. Carta;G. D. Simone;J. Winum;C. T. Supuran (2012). Development of potent carbonic anhydrase inhibitors incorporating both sulfonamide and sulfamide groups.. JOURNAL OF MEDICINAL CHEMISTRY, vol. 55, pp. 6776-6783, ISSN:0022-2623 DOI   Accesso ONLINE all'editore

  M. Bozdag;T. Dreker;C. Henry;P. Tosco;M. Vallaro;R. Fruttero;A. Scozzafava;F. Carta;C. T. Supuran (2012). Novel small molecule protein arginine deiminase 4 (PAD4) inhibitors.. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 23, pp. 715-719, ISSN:0960-894X Accesso ONLINE all'editore

  F. Carta;M. Aggarwal;A. Maresca;A. Scozzafava;R. McKenna;E. Masini;C. T. Supuran (2012). Dithiocarbamates strongly inhibit carbonic anhydrases and show antiglaucoma action in vivo.. JOURNAL OF MEDICINAL CHEMISTRY, vol. 55, pp. 1721-1730, ISSN:0022-2623 DOI   Accesso ONLINE all'editore

  F. Carta;A. Maresca;A. Scozzafava;C. T. Supuran (2012). Novel coumarins and 2-thioxo-coumarins as inhibitors of the tumor-associated carbonic anhydrases IX and XII.. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 20, pp. 2266-2273, ISSN:0968-0896 DOI   Accesso ONLINE all'editore

  S. M. Monti;A. Maresca;F. Viparelli;F. Carta;G. D. Simone;F. A. Mühlschlegel;A. Scozzafava;C. T. Supuran (2012). Dithiocarbamates are strong inhibitors of the beta-class fungal carbonic anhydrases from Cryptococcus neoformans, Candida albicans and Candida glabrata.. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 22, pp. 859-862, ISSN:0960-894X DOI   Accesso ONLINE all'editore

  F. Carta;C. T. Supuran;A. Scozzafava (2012). Novel therapies for glaucoma: a patent review 2007 - 2011.. EXPERT OPINION ON THERAPEUTIC PATENTS, vol. 22, pp. 79-88, ISSN:1354-3776 DOI   Accesso ONLINE all'editore

  S. Avram;A. L. Milac;F. Carta;C. T. Supuran (2012). More effective dithiocarbamate derivatives inhibiting carbonic anhydrases, generated by QSAR and computational design.. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 28, pp. 350-359, ISSN:1475-6366 DOI   Accesso ONLINE all'editore

  D. Can;B. Spingler;P. Schmutz;F. Mendes;P. Raposinho;C. Fernandes;F. Carta;A. Innocenti;I. Santos;C. T. Supuran;R. Alberto (2012). [(Cp-R)M(CO)(3) ] (M=Re or (99m) Tc) Arylsulfonamide, Arylsulfamide, and Arylsulfamate Conjugates for Selective Targeting of Human Carbonic Anhydrase IX.. ANGEWANDTE CHEMIE. INTERNATIONAL EDITION, vol. 51, pp. 3354-3357, ISSN:1433-7851 DOI   Accesso ONLINE all'editore

  A. Scozzafava;F. Carta;C. T. Supuran (2012). Secondary and tertiary sulfonamides: a patent review (2008 - 2012).. EXPERT OPINION ON THERAPEUTIC PATENTS, vol. 23, pp. 203-213, ISSN:1354-3776 DOI   Accesso ONLINE all'editore

  F. Carta;M. Aggarwal;A. Maresca;A. Scozzafava;R. McKenna;C. T. Supuran (2012). Dithiocarbamates: a new class of carbonic anhydrase inhibitors. Crystallographic and kinetic investigations.. CHEMICAL COMMUNICATIONS, vol. 48, pp. 1868-1870, ISSN:1359-7345 DOI   Accesso ONLINE all'editore

  F. Allouche;F. Chabchoub;F. Carta;C. T. Supuran (2012). Synthesis of aminocyanopyrazoles via a multi-component reaction and anti-carbonic anhydrase inhibitory activity of their sulfamide derivatives against cytosolic and transmembrane isoforms.. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 28, pp. 343-349, ISSN:1475-6366 DOI   Accesso ONLINE all'editore

  J. Winum;A. Maresca;F. Carta;A. Scozzafava;C. T. Supuran (2012). Polypharmacology of sulfonamides: pazopanib, a multitargeted receptor tyrosine kinase inhibitor in clinical use, potently inhibits several mammalian carbonic anhydrases.. CHEMICAL COMMUNICATIONS, vol. 48, pp. 8177-8179, ISSN:1359-7345 DOI   Accesso ONLINE all'editore

  F. Carta;A. Scozzafava;C. T. Supuran (2012). Sulfonamides: a patent review (2008 - 2012).. EXPERT OPINION ON THERAPEUTIC PATENTS, vol. 22, pp. 747-758, ISSN:1354-3776 DOI   Accesso ONLINE all'editore

  R. G. Gieling;M. Babur;L. Mamnani;N. Burrows;B. A. Telfer;F. Carta;J. Winum;A. Scozzafava;C. T. Supuran;K. J. Williams (2012). Antimetastatic Effect of Sulfamate Carbonic Anhydrase IX Inhibitors in Breast Carcinoma Xenografts.. JOURNAL OF MEDICINAL CHEMISTRY, vol. 55, pp. 5591-5600, ISSN:0022-2623 DOI   Accesso ONLINE all'editore

  L. Dubois;S. Peeters;N. G. Lieuwes;N. Geusens;A. Thiry;S. Wigfield;F. Carta;A. McIntyre;A. Scozzafava;J. Dogné;C. T. Supuran;A. L. Harris;B. Masereel;P. Lambin (2011). Specific inhibition of carbonic anhydrase IX activity enhances the in vivo therapeutic effect of tumor irradiation.. RADIOTHERAPY AND ONCOLOGY, vol. 99, pp. 424-431, ISSN:0167-8140 DOI   Accesso ONLINE all'editore

  A. Maresca;F. Carta;D. Vullo;C. T. Supuran (2011). Dithiocarbamates strongly inhibit the β-class carbonic anhydrases from Mycobacterium tuberculosis.. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, pp. 0-0, ISSN:1475-6366 DOI   Accesso ONLINE all'editore

  N. Pala;R. Dallocchio;A. Dessì;A. Brancale;F. Carta;S. Ihm;A. Maresca;M. Sechi;C. T. Supuran (2011). Virtual screening-driven identification of human carbonic anhydrase inhibitors incorporating an original, new pharmacophore.. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 21, pp. 2515-2520, ISSN:0960-894X DOI   Accesso ONLINE all'editore

  F. Carta;A. Innocenti;R. A. Hall;F. A. Mühlschlegel;A. Scozzafava;C. T. Supuran (2011). Carbonic anhydrase inhibitors. Inhibition of the β-class enzymes from the fungal pathogens Candida albicans and Cryptococcus neoformans with branched aliphatic/aromatic carboxylates and their derivatives.. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 21, pp. 2521-2526, ISSN:0960-894X DOI   Accesso ONLINE all'editore

  Y.Lou; P.C. McDonald; A.Oloumi; S.Chia; C.Ostlund; A. Ahmadi; A.Kyle; U.auf dem Keller; S.Leung; D.Huntsman; B.Clarke; B.W.Sutherland; D.Waterhouse; M.Bally; C.Roskelley; C.M. Overall; A.Minchinton; F.Pacchiano; F. Carta; A.Scozzafava; N.Touisni; J.-Y.Winum; C.T. Supuran; S.Dedhar (2011). Targeting Tumor Hypoxia: Suppression of Breast TumorGrowth and Metastasis by Novel Carbonic Anhydrase IX Inhibitors. CANCER RESEARCH, vol. -----------------, pp. 0-0, ISSN:0008-5472 DOI   Accesso ONLINE all'editore

  F. Carta;V. Garaj;A. Maresca;J. Wagner;B. S. Avvaru;A. H. Robbins;A. Scozzafava;R. McKenna;C. T. Supuran (2011). Sulfonamides incorporating 1,3,5-triazine moieties selectively and potently inhibit carbonic anhydrase transmembrane isoforms IX, XII and XIV over cytosolic isoforms I and II: Solution and X-ray crystallographic studies.. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 19, pp. 3105-3119, ISSN:0968-0896 DOI   Accesso ONLINE all'editore

  claudiu supuran, andrea scozzafava, fabrizio carta (2011). CARBONIC ANHYDRASE INHIBITOR COMPRISING A DITHIOCARBAMATE. Numero: WO2013050426 (A1) SUPURAN CLAUDIU T [IT]; SCOZZAFAVA ANDREA [IT]; MASINI EMANUELA [IT]; CARTA FABRIZIO [IT]; PETTERSEN ERIK OLAI [NO]; EBBESEN PETER [DK]

  F. Pacchiano;F. Carta;D. Vullo;A. Scozzafava;C. T. Supuran (2011). Inhibition of β-carbonic anhydrases with ureido-substituted benzenesulfonamides.. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 21, pp. 102-105, ISSN:0960-894X DOI   Accesso ONLINE all'editore

  F. Pacchiano; F. Carta; P.C. McDonald; Y. Lou; D.Vullo; A. Scozzafava; S. Dedhar; and C.T. Supuran (2011). Ureido-Substituted Benzenesulfonamides Potently Inhibit Carbonic Anhydrase IX and Show Antimetastatic Activity in a Model of Breast Cancer Metastasis. JOURNAL OF MEDICINAL CHEMISTRY, vol. 54, pp. 1896-1902, ISSN:0022-2623 DOI   Accesso ONLINE all'editore

  F. Carta;C. Temperini;A. Innocenti;A. Scozzafava;K. Kaila;C. T. Supuran (2010). Polyamines inhibit carbonic anhydrases by anchoring to the zinc-coordinated water molecule.. JOURNAL OF MEDICINAL CHEMISTRY, vol. 53, pp. 5511-5522, ISSN:1520-4804 DOI   Accesso ONLINE all'editore

  Alder, Roger W.*; Carta, Fabrizio; Reed, Christopher A.; Stoyanova, Irina; Willis, Christine L. (2010). Searching for intermediates in Prins cyclisations: The 2-oxa-5-adamantyl carbocation. ORGANIC & BIOMOLECULAR CHEMISTRY, vol. 8, pp. 1551-1559, ISSN:1477-0520 DOI  

  I. Nishimori;T. Minakuchi;A. Maresca;F. Carta;A. Scozzafava;C. T. Supuran (2010). The β-carbonic anhydrases from Mycobacterium tuberculosis as drug targets.. CURRENT PHARMACEUTICAL DESIGN, vol. 16, pp. 3300-3309, ISSN:1381-6128

  SUPURAN CLAUDIU, DEDHAR SHOUKAT, CARTA FABRIZIO, WINUM JEAN-YVES, MCDONALD PAUL C (2010). CARBONIC ANHYDRASE INHIBITORS WITH ANTIMETASTATIC ACTIVITY. Numero: WO2012070024 (A1) SUPURAN CLAUDIU [IT]; DEDHAR SHOUKAT [CA]; CARTA FABRIZIO [IT]; WINUM JEAN-YVES [FR]; MCDONALD PAUL C [CA]

  SUPURAN CLAUDIU; DEDHAR SHOUKAT; MCDONALD PAUL; CARTA FABRIZIO (2010). NOVEL SULFONAMIDE COMPOUNDS FOR INHIBITION OF METASTATIC TUMOR GROWTH. Numero: WO2012021963 (A1) SUPURAN CLAUDIU; DEDHAR SHOUKAT; MCDONALD PAUL; CARTA FABRIZIO

  A. Maresca;F. Carta;D. Vullo;A. Scozzafava;C. T. Supuran (2009). Carbonic anhydrase inhibitors. Inhibition of the Rv1284 and Rv3273 beta-carbonic anhydrases from Mycobacterium tuberculosis with diazenylbenzenesulfonamides.. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 19, pp. 4929-4932, ISSN:0960-894X DOI   Accesso ONLINE all'editore

  F. Carta;B. Pothen;A. Maresca;M. Tiwari;V. Singh;C. T. Supuran (2009). Carbonic anhydrase inhibitors: inhibition of cytosolic carbonic anhydrase isozymes II and VII with simple aromatic sulfonamides and some azo dyes.. CHEMICAL BIOLOGY & DRUG DESIGN, vol. 74, pp. 196-202, ISSN:1747-0285 DOI   Accesso ONLINE all'editore

  Sechi, M; Carta, F; Sannia, L; Dallocchio, R; Dessi, A; Al-Safi, RI; Neamati, N (2009). Design, synthesis, molecular modeling, and anti-HIV-1 integrase activity of a series of photoactivatable diketo acid-containing inhibitors as affinity probes. ANTIVIRAL RESEARCH, vol. 81, pp. 267-276, ISSN:0166-3542 DOI  

  F. Carta;A. Maresca;A. Scozzafava;D. Vullo;C. T. Supuran (2009). Carbonic anhydrase inhibitors. Diazenylbenzenesulfonamides are potent and selective inhibitors of the tumor-associated isozymes IX and XII over the cytosolic isoforms I and II.. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 17, pp. 7093-7099, ISSN:0968-0896 DOI   Accesso ONLINE all'editore

  F. Carta;A. Maresca;A. S. Covarrubias;S. L. Mowbray;T. A. Jones;C. T. Supuran (2009). Carbonic anhydrase inhibitors. Characterization and inhibition studies of the most active beta-carbonic anhydrase from Mycobacterium tuberculosis, Rv3588c.. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 19, pp. 6649-6654, ISSN:0960-894X DOI   Accesso ONLINE all'editore

  Bacchi, Alessia; Biemmi, Mariano; Carcelli, Mauro; Carta, Fabrizio; Compari, Carlotta; Fisicaro, Emilia; Rogolino, Dominga; Sechi, Mario*; Sippel, Martin; Sotriffer, Christoph A.; Sanchez, Tino W.; Neamati, Nouri (2008). From ligand to complexes. Part 2. Remarks on human immunodeficiency virus type 1 integrase inhibition by β-diketo acid metal complexes. JOURNAL OF MEDICINAL CHEMISTRY, vol. 51, pp. 7253-7264, ISSN:0022-2623 DOI  

  Sechi, Mario*; Sannia, Luciano; Carta, Fabrizio; Palomba, Michele; Dallocchio, Roberto; Dessì, Alessandro; Derudas, Massimiliano; Zawahir, Zahrah; Neamati, Nouri (2005). Design of novel bioisosteres of β-diketo acid inhibitors of HIV-1 integrase. ANTIVIRAL CHEMISTRY & CHEMOTHERAPY, vol. 16, pp. 41-61, ISSN:0956-3202 DOI   Accesso ONLINE all'editore

  Sechi, Mario*; Derudas, Massimiliano; Dallocchio, Roberto; Dessì, Alessandro; Bacchi, Alessia; Sannia, Luciano; Carta, Fabrizio; Palomba, Michele; Ragab, Omar; Chan, Carney; Shoemaker, Robert; Sei, Shizuko; Dayam, Raveendra; Neamati, Nouri (2004). Design and synthesis of novel indole β-diketo acid derivatives as HIV-1 integrase inhibitors. JOURNAL OF MEDICINAL CHEMISTRY, vol. 47, pp. 5298-5310, ISSN:0022-2623 DOI  

  Sechi, Mario*; Angotzi, Gianfranco; Dallocchio, Roberto; Dessi, Alessandro; Carta, Fabrizio; Sannia, Luciano; Mariani, Alberto; Fiori, Stefano; Sanchez, Tino; Movsessian, Leah; Plasencia, Carmen; Neamati, Nouri (2004). Design and synthesis of novel dihydroxyindole-2-carboxylic acids as HIV-1 integrase inhibitors. ANTIVIRAL CHEMISTRY & CHEMOTHERAPY, vol. 15, pp. 67-81, ISSN:0956-3202 DOI   Accesso ONLINE all'editore

  Sechi, Mario; Sannia, Luciano; Orecchioni, Maria; Carta, Fabrizio; Paglietti, Giuseppe; Neamati, Nouri (2003). Structural Investigation of 3,5-Disubstituted Isoxazoles by1H-Nuclear Magnetic Resonance. JOURNAL OF HETEROCYCLIC CHEMISTRY, vol. 40, pp. 1097-1102, ISSN:0022-152X DOI   Accesso ONLINE all'editore